Myosin Kinase Inhibiting Peptide
CAS No. 119386-39-9
Myosin Kinase Inhibiting Peptide ( ——— )
产品货号. M41241 CAS No. 119386-39-9
Myosin light chain kinase fragment 11-19 amide (MLCK(11-19) amide) 是 MLCK 的底物特异性多肽抑制剂。Myosin light chain kinase fragment 11-19 amide 可抑制低渗诱导的 Ca2+ 进入细胞。Myosin light chain kinase fragment 11-19 amide 可用于人类宫颈癌的研究。
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 25MG | 获取报价 | 有现货 |
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| 50MG | 获取报价 | 有现货 |
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| 100MG | 获取报价 | 有现货 |
|
生物学信息
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产品名称Myosin Kinase Inhibiting Peptide
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述Myosin light chain kinase fragment 11-19 amide (MLCK(11-19) amide) 是 MLCK 的底物特异性多肽抑制剂。Myosin light chain kinase fragment 11-19 amide 可抑制低渗诱导的 Ca2+ 进入细胞。Myosin light chain kinase fragment 11-19 amide 可用于人类宫颈癌的研究。
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产品描述Myosin light chain kinase fragment 11-19 amide (MLCK(11-19) amide) is a substrate-specific peptide inhibitor of MLCK. Myosin light chain kinase fragment 11-19 amide inhibits hypotonicity-induced Ca2+ entry. Myosin light chain kinase fragment 11-19 amide can be used in the research of human cervical cancer.
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体外实验———
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体内实验Myosin light chain kinase fragment 11-19 amide (5 μM) reduces the amplitude and rate of activation of noradrenaline-evoked non-selective cation current (Icat) in rabbit portal vein myocytes.Myosin light chain kinase fragment 11-19 amide inhibits swelling-activated taurine transport with an IC50 value of 2.0 μM.Myosin light chain kinase fragment 11-19 amide (10 μM) inhibits β2-integrin-mediated adhesion in neutrophils treated with KT5720 (25 μM).
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同义词———
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通路Others
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靶点Other Targets
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受体MLCK
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研究领域———
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适应症———
化学信息
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CAS Number119386-39-9
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分子量987.2
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分子式C40H78N18O11
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纯度>98% (HPLC)
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溶解度———
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SMILES———
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化学全称———
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Aromolaran AS, et al. Evidence for myosin light chain kinase mediating noradrenaline-evoked cation current in rabbit portal vein myocytes. J Physiol. 2000 May 1;524 Pt 3(Pt 3):853-63. ?
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